| Year |
Citation |
Score |
| 2020 |
Bagnolini G, Milano D, Manerba M, Schipani F, Ortega JA, Gioia D, Falchi F, Balboni A, Farabegoli F, De Franco F, Robertson J, Pellicciari R, Pallavicini I, Peri S, Minucci S, ... ... Roberti M, et al. Synthetic lethality in pancreatic cancer: discovery of a new RAD51-BRCA2 small molecule disruptor that inhibits homologous recombination and synergizes with olaparib. Journal of Medicinal Chemistry. PMID 32037829 DOI: 10.1021/Acs.Jmedchem.9B01526 |
0.557 |
|
| 2020 |
Linciano P, Cullia G, Borsari C, Santucci M, Ferrari S, Witt G, Gul S, Kuzikov M, Ellinger B, Santarém N, Cordeiro da Silva A, Conti P, Bolognesi ML, Roberti M, Prati F, et al. Identification of a 2,4-diaminopyrimidine scaffold targeting Trypanosoma brucei pteridine reductase 1 from the LIBRA compound library screening campaign. European Journal of Medicinal Chemistry. 189: 112047. PMID 31982652 DOI: 10.1016/J.Ejmech.2020.112047 |
0.446 |
|
| 2019 |
Roberti M, Schipani F, Bagnolini G, Milano D, Giacomini E, Falchi F, Balboni A, Manerba M, Farabegoli F, De Franco F, Robertson J, Minucci S, Pallavicini I, Di Stefano G, Girotto S, et al. Rad51/BRCA2 disruptors inhibit homologous recombination and synergize with olaparib in pancreatic cancer cells. European Journal of Medicinal Chemistry. 165: 80-92. PMID 30660828 DOI: 10.1016/J.Ejmech.2019.01.008 |
0.532 |
|
| 2018 |
Uliassi E, Peña-Altamira LE, Morales AV, Massenzio F, Petralla S, Rossi M, Roberti M, Martínez-González L, Martínez A, Monti B, Bolognesi ML. A focused library of psychotropic analogs with neuroprotective and neuroregenerative potential. Acs Chemical Neuroscience. PMID 30253086 DOI: 10.1021/Acschemneuro.8B00242 |
0.391 |
|
| 2018 |
Porru E, Franco P, Calabria D, Spinozzi S, Roberti M, Caliceti C, Roda A. Combined analytical approaches to define biodistribution and biological activity of semi-synthetic berberrubine, the active metabolite of natural berberine. Analytical and Bioanalytical Chemistry. PMID 29411090 DOI: 10.1007/S00216-018-0884-2 |
0.326 |
|
| 2017 |
Bruno F, Castelli G, Vitale F, Giacomini E, Roberti M, Colomba C, Cascio A, Tolomeo M. Effects of trans-stilbene and terphenyl compounds on different strains of Leishmania and on cytokines production from infected macrophages. Experimental Parasitology. PMID 29154845 DOI: 10.1016/J.Exppara.2017.11.004 |
0.301 |
|
| 2017 |
Falchi F, Giacomini E, Masini T, Boutard N, Di Ianni L, Manerba M, Farabegoli F, Rossini L, Robertson J, Minucci S, Pallavicini I, Di Stefano G, Pellicciari R, Roberti M, Cavalli A. Synthetic lethality triggered by combining Olaparib with BRCA2-Rad51 disruptors. Acs Chemical Biology. PMID 28841282 DOI: 10.1021/Acschembio.7B00707 |
0.551 |
|
| 2017 |
Manerba M, Di Ianni L, Govoni M, Roberti M, Recanatini M, Di Stefano G. LDH inhibition impacts on heat shock response and induces senescence of hepatocellular carcinoma cells. European Journal of Pharmaceutical Sciences : Official Journal of the European Federation For Pharmaceutical Sciences. 105: 91-98. PMID 28501492 DOI: 10.1016/J.Ejps.2017.05.015 |
0.35 |
|
| 2016 |
Jeřábek J, Uliassi E, Guidotti L, Korábečný J, Soukup O, Sepsova V, Hrabinova M, Kuča K, Bartolini M, Peña-Altamira LE, Petralla S, Monti B, Roberti M, Bolognesi ML. Tacrine-resveratrol fused hybrids as multi-target-directed ligands against Alzheimer's disease. European Journal of Medicinal Chemistry. 127: 250-262. PMID 28064079 DOI: 10.1016/J.Ejmech.2016.12.048 |
0.358 |
|
| 2016 |
Rupiani S, Guidotti L, Manerba M, Ianni LD, Giacomini E, Falchi F, Stefano GD, Roberti M, Recanatini M. Synthesis of natural urolithin M6, a galloflavin mimetic, as a potential inhibitor of lactate dehydrogenase A. Organic & Biomolecular Chemistry. PMID 27827510 DOI: 10.1039/C6Ob01977C |
0.734 |
|
| 2016 |
Manerba M, Di Ianni L, Govoni M, Roberti M, Recanatini M, Di Stefano G. Lactate dehydrogenase inhibitors can reverse inflammation induced changes in colon cancer cells. European Journal of Pharmaceutical Sciences : Official Journal of the European Federation For Pharmaceutical Sciences. PMID 27622920 DOI: 10.1016/J.Ejps.2016.09.014 |
0.385 |
|
| 2016 |
Giacomini E, Rupiani S, Guidotti L, Recanatini M, Roberti M. The Use of Stilbene Scaffold in Medicinal Chemistry and Multi-Target Drug Design. Current Medicinal Chemistry. PMID 27183980 DOI: 10.2174/0929867323666160517121629 |
0.727 |
|
| 2016 |
Garuti L, Roberti M, Bottegoni G, Ferraro M. Diaryl Urea: a Privileged Structure in Anticancer Agents. Current Medicinal Chemistry. PMID 27063259 DOI: 10.2174/0929867323666160411142532 |
0.425 |
|
| 2016 |
Castelli G, Bruno F, Vitale F, Roberti M, Colomba C, Giacomini E, Guidotti L, Cascio A, Tolomeo M. In vitro Antileishmanial Activity of trans-Stilbene and Terphenyl Compounds. Experimental Parasitology. PMID 26953250 DOI: 10.1016/J.Exppara.2016.03.007 |
0.424 |
|
| 2015 |
Rupiani S, Buonfiglio R, Manerba M, Di Ianni L, Vettraino M, Giacomini E, Masetti M, Falchi F, Di Stefano G, Roberti M, Recanatini M. Identification of N-acylhydrazone derivatives as novel lactate dehydrogenase A inhibitors. European Journal of Medicinal Chemistry. 101: 63-70. PMID 26114812 DOI: 10.1016/J.Ejmech.2015.06.028 |
0.75 |
|
| 2015 |
Manerba M, Di Ianni L, Fiume L, Roberti M, Recanatini M, Di Stefano G. Lactate dehydrogenase inhibitors sensitize lymphoma cells to cisplatin without enhancing the drug effects on immortalized normal lymphocytes. European Journal of Pharmaceutical Sciences : Official Journal of the European Federation For Pharmaceutical Sciences. 74: 95-102. PMID 25930121 DOI: 10.1016/J.Ejps.2015.04.022 |
0.406 |
|
| 2015 |
Giacomini E, Buonfiglio R, Masetti M, Wang Y, Tseng GN, Roberti M, Recanatini M. A ligand-based virtual screening approach to identify small molecules as HERG channel activators. Combinatorial Chemistry & High Throughput Screening. 18: 269-80. PMID 25747449 DOI: 10.2174/1386207318666150305121841 |
0.389 |
|
| 2015 |
Garuti L, Roberti M, Bottegoni G. Multi-kinase inhibitors. Current Medicinal Chemistry. 22: 695-712. PMID 25511779 DOI: 10.2174/0929867321666141216125528 |
0.397 |
|
| 2015 |
Rupiani S, Buonfiglio R, Manerba M, Di Ianni L, Vettraino M, Giacomini E, Masetti M, Falchi F, Di Stefano G, Roberti M, Recanatini M. Identification of N-acylhydrazone derivatives as novel lactate dehydrogenase A inhibitors European Journal of Medicinal Chemistry. 101: 63-70. DOI: 10.1016/j.ejmech.2015.06.028 |
0.717 |
|
| 2014 |
Nepovimova E, Uliassi E, Korabecny J, Peña-Altamira LE, Samez S, Pesaresi A, Garcia GE, Bartolini M, Andrisano V, Bergamini C, Fato R, Lamba D, Roberti M, Kuca K, Monti B, et al. Multitarget drug design strategy: Quinone-tacrine hybrids designed to block amyloid-β aggregation and to exert anticholinesterase and antioxidant effects Journal of Medicinal Chemistry. 57: 8576-8589. PMID 25259726 DOI: 10.1021/Jm5010804 |
0.379 |
|
| 2014 |
Giacomini E, Nebbioso A, Ciotta A, Ianni C, Falchi F, Roberti M, Tolomeo M, Grimaudo S, Cristina AD, Pipitone RM, Altucci L, Recanatini M. Novel antiproliferative chimeric compounds with marked histone deacetylase inhibitory activity. Acs Medicinal Chemistry Letters. 5: 973-8. PMID 25221651 DOI: 10.1021/Ml5000959 |
0.469 |
|
| 2014 |
Spinozzi S, Colliva C, Camborata C, Roberti M, Ianni C, Neri F, Calvarese C, Lisotti A, Mazzella G, Roda A. Berberine and its metabolites: Relationship between physicochemical properties and plasma levels after administration to human subjects Journal of Natural Products. 77: 766-772. PMID 24593257 DOI: 10.1021/Np400607K |
0.305 |
|
| 2014 |
Garuti L, Roberti M, Bottegoni G. Benzimidazole derivatives as kinase inhibitors Current Medicinal Chemistry. 21: 2284-2298. PMID 24533813 DOI: 10.2174/0929867321666140217105714 |
0.39 |
|
| 2013 |
Turroni S, Tolomeo M, Mamone G, Picariello G, Giacomini E, Brigidi P, Roberti M, Grimaudo S, Pipitone RM, Di Cristina A, Recanatini M. A Natural-Like Synthetic Small Molecule Impairs Bcr-Abl Signaling Cascades and Induces Megakaryocyte Differentiation in Erythroleukemia Cells Plos One. 8. PMID 23460890 DOI: 10.1371/Journal.Pone.0057650 |
0.361 |
|
| 2013 |
Tolomeo M, Roberti M, Scapozza L, Tarantelli C, Giacomini E, Titone L, Saporito L, Di Carlo P, Colomba C. TTAS a new stilbene derivative that induces apoptosis in Leishmania infantum Experimental Parasitology. 133: 37-43. PMID 23103597 DOI: 10.1016/J.Exppara.2012.10.006 |
0.408 |
|
| 2012 |
Farabegoli F, Vettraino M, Manerba M, Fiume L, Roberti M, Di Stefano G. Galloflavin, a new lactate dehydrogenase inhibitor, induces the death of human breast cancer cells with different glycolytic attitude by affecting distinct signaling pathways European Journal of Pharmaceutical Sciences. 47: 729-738. PMID 22954722 DOI: 10.1016/J.Ejps.2012.08.012 |
0.36 |
|
| 2012 |
Cavalli A, Buonfiglio R, Ianni C, Masetti M, Ceccarini L, Caves R, Chang MWY, Mitcheson JS, Roberti M, Recanatini M. Computational design and discovery of "minimally structured" hERG blockers Journal of Medicinal Chemistry. 55: 4010-4014. PMID 22455383 DOI: 10.1021/Jm201194Q |
0.378 |
|
| 2012 |
Chiriano G, De Simone A, Mancini F, Perez DI, Cavalli A, Bolognesi ML, Legname G, Martinez A, Andrisano V, Carloni P, Roberti M. A small chemical library of 2-aminoimidazole derivatives as BACE-1 inhibitors: Structure-based design, synthesis, and biological evaluation. European Journal of Medicinal Chemistry. 48: 206-13. PMID 22209418 DOI: 10.1016/J.Ejmech.2011.12.016 |
0.443 |
|
| 2012 |
Manerba M, Vettraino M, Fiume L, di Stefano G, Sartini A, Giacomini E, Buonfiglio R, Roberti M, Recanatini M. Galloflavin (CAS 568-80-9): A Novel Inhibitor of Lactate Dehydrogenase Chemmedchem. 7: 311-317. PMID 22052811 DOI: 10.1002/Cmdc.201100471 |
0.431 |
|
| 2011 |
Garuti L, Roberti M, Bottegoni G. Irreversible protein kinase inhibitors Current Medicinal Chemistry. 18: 2981-2994. PMID 21651479 DOI: 10.2174/092986711796391705 |
0.425 |
|
| 2011 |
Chiriano G, Sartini A, Mancini F, Andrisano V, Bolognesi ML, Roberti M, Recanatini M, Carloni P, Cavalli A. Sequential virtual screening approach to the identification of small organic molecules as potential BACE-1 inhibitors. Chemical Biology & Drug Design. 77: 268-71. PMID 21244641 DOI: 10.1111/J.1747-0285.2011.01087.X |
0.374 |
|
| 2010 |
Bongarzone S, Tran HNA, Cavalli A, Roberti M, Carloni P, Legname G, Bolognesi ML. Parallel synthesis, evaluation, and preliminary structure-activity relationship of 2,5-diamino-1,4-benzoquinones as a novel class of bivalent anti-prion compound Journal of Medicinal Chemistry. 53: 8197-8201. PMID 21047125 DOI: 10.1021/Jm100882T |
0.394 |
|
| 2010 |
Garuti L, Roberti M, Bottegoni G. Non-ATP competitive protein kinase inhibitors Current Medicinal Chemistry. 17: 2804-2821. PMID 20586715 DOI: 10.2174/092986710791859333 |
0.358 |
|
| 2010 |
Roberti M, Natalini B, Andrisano V, Seraglia R, Gioiello A, Pellicciari R. Thermal and catalytic reactions of ethyl diazopyruvate with [60]fullerene Tetrahedron. 66: 7329-7332. DOI: 10.1016/J.Tet.2010.06.067 |
0.473 |
|
| 2009 |
Pizzirani D, Roberti M, Grimaudo S, Di Cristina A, Pipitone RM, Tolomeo M, Recanatini M. Identification of biphenyl-based hybrid molecules able to decrease the intracellular level of Bcl-2 protein in Bcl-2 overexpressing leukemia cells Journal of Medicinal Chemistry. 52: 6936-6940. PMID 19764793 DOI: 10.1021/Jm900907S |
0.426 |
|
| 2009 |
Garuti L, Roberti M, Bottegoni G. Small molecule Aurora kinases inhibitors Current Medicinal Chemistry. 16: 1949-1963. PMID 19519375 DOI: 10.2174/092986709788682227 |
0.424 |
|
| 2008 |
Garuti L, Roberti M, Pizzirani D. Synthetic small molecule Cdc25 phosphatases inhibitors Current Medicinal Chemistry. 15: 573-580. PMID 18336271 DOI: 10.2174/092986708783769722 |
0.496 |
|
| 2008 |
Pizzirani D, Roberti M, Cavalli A, Grimaudo S, Di Cristina A, Pipitone RM, Gebbia N, Tolomeo M, Recanatini M. Antiproliferative agents that interfere with the cell cycle at the G 1→S transition: Further development and characterization of a small library of stilbene-derived compounds Chemmedchem. 3: 345-355. PMID 18161738 DOI: 10.1002/Cmdc.200700258 |
0.442 |
|
| 2007 |
Garuti L, Roberti M, Pizzirani D. Nitrogen-containing heterocyclic quinones: A class of potential selective antitumor agents Mini-Reviews in Medicinal Chemistry. 7: 481-489. PMID 17504183 DOI: 10.2174/138955707780619626 |
0.404 |
|
| 2007 |
Kaur G, Roberti M, Raul F, Pendurthi UR. Suppression of human monocyte tissue factor induction by red wine phenolics and synthetic derivatives of resveratrol. Thrombosis Research. 119: 247-56. PMID 16507316 DOI: 10.1016/J.Thromres.2006.01.020 |
0.356 |
|
| 2007 |
Pizzirani D, Roberti M, Recanatini M. Domino Knoevenagel/Diels-Alder sequence coupled to Suzuki reaction: a valuable synthetic platform for chemical biology Tetrahedron Letters. 48: 7120-7124. DOI: 10.1016/J.Tetlet.2007.07.214 |
0.301 |
|
| 2006 |
Roberti M, Pizzirani D, Recanatini M, Simoni D, Grimaudo S, Di Cristina A, Abbadessa V, Gebbia N, Tolomeo M. Identification of a terphenyl derivative that blocks the cell cycle in the G0-G1 phase and induces differentiation in leukemia cells. Journal of Medicinal Chemistry. 49: 3012-8. PMID 16686543 DOI: 10.1021/Jm060253O |
0.361 |
|
| 2006 |
Simoni D, Roberti M, Invidiata FP, Aiello E, Aiello S, Marchetti P, Baruchello R, Eleopra M, Di Cristina A, Grimaudo S, Gebbia N, Crosta L, Dieli F, Tolomeo M. Stilbene-based anticancer agents: resveratrol analogues active toward HL60 leukemic cells with a non-specific phase mechanism. Bioorganic & Medicinal Chemistry Letters. 16: 3245-8. PMID 16580204 DOI: 10.1016/J.Bmcl.2006.03.028 |
0.379 |
|
| 2005 |
Simoni D, Giannini G, Roberti M, Rondanin R, Baruchello R, Rossi M, Grisolia G, Invidiata FP, Aiello S, Marino S, Cavallini S, Siniscalchi A, Gebbia N, Crosta L, Grimaudo S, et al. Studies on the apoptotic activity of natural and synthetic retinoids: discovery of a new class of synthetic terphenyls that potently support cell growth and inhibit apoptosis in neuronal and HL-60 cells. Journal of Medicinal Chemistry. 48: 4293-9. PMID 15974583 DOI: 10.1021/Jm049080Y |
0.382 |
|
| 2005 |
Tolomeo M, Grimaudo S, Di Cristina A, Roberti M, Pizzirani D, Meli M, Dusonchet L, Gebbia N, Abbadessa V, Crosta L, Barucchello R, Grisolia G, Invidiata F, Simoni D. Pterostilbene and 3'-hydroxypterostilbene are effective apoptosis-inducing agents in MDR and BCR-ABL-expressing leukemia cells. The International Journal of Biochemistry & Cell Biology. 37: 1709-26. PMID 15878840 DOI: 10.1016/J.Biocel.2005.03.004 |
0.379 |
|
| 2005 |
Simoni D, Rossi M, Bertolasi V, Roberti M, Pizzirani D, Rondanin R, Baruchello R, Invidiata FP, Tolomeo M, Grimaudo S, Merighi S, Varani K, Gessi S, Borea PA, Marino S, et al. Synthesis and pharmacology of 6-substituted benztropines: discovery of novel dopamine uptake inhibitors possessing low binding affinity to the dopamine transporter. Journal of Medicinal Chemistry. 48: 3337-43. PMID 15857139 DOI: 10.1021/Jm0490235 |
0.318 |
|
| 2005 |
Simoni D, Grisolia G, Giannini G, Roberti M, Rondanin R, Piccagli L, Baruchello R, Rossi M, Romagnoli R, Invidiata FP, Grimaudo S, Jung MK, Hamel E, Gebbia N, Crosta L, et al. Heterocyclic and phenyl double-bond-locked combretastatin analogues possessing potent apoptosis-inducing activity in HL60 and in MDR cell lines. Journal of Medicinal Chemistry. 48: 723-36. PMID 15689156 DOI: 10.1021/Jm049622B |
0.37 |
|
| 2005 |
Grimaudo S, Di Cristina A, Abbadessa V, Daniele S, Roberti M, Tolomeo M. Novel Stilbene-Based Antileukemic Agents Active in P-Glycoprotein Expressing and Apoptosis-Resistant Acute Leukaemia Cell Lines. Blood. 106: 4436-4436. DOI: 10.1182/Blood.V106.11.4436.4436 |
0.428 |
|
| 2004 |
Chatgilialoglu C, Ferreri C, Gimisis T, Roberti M, Balzarini J, De Clercq E. Synthesis and biological evaluation of novel 1'-branched and spironucleoside analogues. Nucleosides, Nucleotides & Nucleic Acids. 23: 1565-81. PMID 15620096 DOI: 10.1081/Ncn-200031391 |
0.428 |
|
| 2004 |
Garuti L, Roberti M, Pizzirani D, Pession A, Leoncini E, Cenci V, Hrelia S. Differential antiproliferative activity of new benzimidazole-4,7-diones. Farmaco (Società Chimica Italiana : 1989). 59: 663-8. PMID 15262537 DOI: 10.1016/J.Farmac.2004.04.001 |
0.406 |
|
| 2003 |
Roberti M, Pizzirani D, Simoni D, Rondanin R, Baruchello R, Bonora C, Buscemi F, Grimaudo S, Tolomeo M. Synthesis and biological evaluation of resveratrol and analogues as apoptosis-inducing agents. Journal of Medicinal Chemistry. 46: 3546-54. PMID 12877593 DOI: 10.1021/Jm030785U |
0.419 |
|
| 2002 |
Garuti L, Roberti M, De Clercq E. Synthesis and antiviral/antiproliferative activity of some N-sulphonylbenzimidazoles. Bioorganic & Medicinal Chemistry Letters. 12: 2707-10. PMID 12217359 DOI: 10.1016/S0960-894X(02)00535-8 |
0.421 |
|
| 2001 |
Garuti L, Roberti M, Gentilomi G. Synthesis and antiviral assays of some benzimidazole nucleosides and acyclonucleosides Farmaco. 56: 815-819. PMID 11765032 DOI: 10.1016/S0014-827X(01)01164-8 |
0.382 |
|
| 2001 |
Garuti L, Roberti M, Pession A, Leoncini E, Hrelia S. Synthesis and antiproliferative activity of some thiazolylbenzimidazole-4,7-diones Bioorganic and Medicinal Chemistry Letters. 11: 3147-3149. PMID 11720862 DOI: 10.1016/S0960-894X(01)00639-4 |
0.389 |
|
| 2001 |
Simoni D, Roberti M, Invidiata FP, Rondanin R, Baruchello R, Malagutti C, Mazzali A, Rossi M, Grimaudo S, Capone F, Dusonchet L, Meli M, Raimondi MV, Landino M, D'Alessandro N, et al. Heterocycle-containing retinoids. Discovery of a novel isoxazole arotinoid possessing potent apoptotic activity in multidrug and drug-induced apoptosis-resistant cells Journal of Medicinal Chemistry. 44: 2308-2318. PMID 11428925 DOI: 10.1021/Jm0010320 |
0.384 |
|
| 2001 |
Simoni D, Roberti M, Rondanin R, Baruchello R, Rossi M, Invidiata FP, Merighi S, Varani K, Gessi S, Borea PA, Marino S, Cavallini S, Bianchi C, Siniscalchi A. Effects of two-carbon bridge region methoxylation of benztropine: Discovery of novel chiral ligands for the dopamine transporter Bioorganic and Medicinal Chemistry Letters. 11: 823-827. PMID 11277529 DOI: 10.1016/S0960-894X(01)00068-3 |
0.302 |
|
| 2001 |
Simoni D, Rondanin R, Baruchello R, Roberti M, Rossi M, Grimaudo S, D'Alessandro N, Invidiata FP, Tolomeo M. Retinoic acid and analogs as potent inducers of differentiation and apoptosis. New promising chemopreventive and chemotherapeutic agents in oncology Pure and Applied Chemistry. 73: 1437-1444. DOI: 10.1351/Pac200173091437 |
0.418 |
|
| 2000 |
Simoni D, Roberti M, Paolo Invidiata F, Rondanin R, Baruchello R, Malagutti C, Mazzali A, Rossi M, Grimaudo S, Dusonchet L, Meli M, Raimondi MV, D'Alessandro N, Tolomeo M. Programmed cell death (PCD) associated with the stilbene motif of arotinoids: Discovery of novel apoptosis inducer agents possessing activity on multidrug resistant tumor cells Bioorganic and Medicinal Chemistry Letters. 10: 2669-2673. PMID 11128648 DOI: 10.1016/S0960-894X(00)00547-3 |
0.378 |
|
| 2000 |
Garuti L, Roberti M, Malagoli M, Rossi T, Castelli M. Synthesis and antiproliferative activity of some benzimidazole-4,7-dione derivatives Bioorganic and Medicinal Chemistry Letters. 10: 2193-2195. PMID 11012027 DOI: 10.1016/S0960-894X(00)00429-7 |
0.401 |
|
| 2000 |
Garuti L, Roberti M, Gentilomi G. Synthesis and antiviral assays of some 2-substituted benzimidazole-N- carbamates Farmaco. 55: 35-39. PMID 10755229 DOI: 10.1016/S0014-827X(99)00117-2 |
0.384 |
|
| 2000 |
Roberti M, Rondanin R, Ferroni R, Baruchello R, Invidiata FP, Andrisano V, Bertucci C, Bertolasi V, Grimaudo S, Tolomeo M, Simoni D. Pig liver esterase (PLE)-mediated resolution of N-substituted 4-benzoyloxy-3-carbomethoxypiperidines: A convenient preparation of 4-hydroxy- and 4-benzoyloxy-3-carbomethoxypiperidines in enantiomerically pure form Tetrahedron Asymmetry. 11: 4397-4405. DOI: 10.1016/S0957-4166(00)00404-3 |
0.323 |
|
| 1999 |
Garuti L, Roberti M, Cermelli C. Synthesis and antiviral activity of some N-benzenesulphonylbenzimidazoles Bioorganic and Medicinal Chemistry Letters. 9: 2525-2530. PMID 10498201 DOI: 10.1016/S0960-894X(99)00429-1 |
0.365 |
|
| 1999 |
Simoni D, Roberti M, Andrisano V, Manferdini M, Rondanin R, Invidiata FP. Two-carbon bridge substituted cocaines: Enantioselective synthesis, attribution of the absolute configuration and biological activity of novel 6- and 7-methoxylated cocaines Farmaco. 54: 275-287. PMID 10418122 DOI: 10.1016/S0014-827X(99)00027-0 |
0.336 |
|
| 1999 |
Kozikowski AP, Simoni D, Roberti M, Rondanin R, Wang S, Du P, Johnson KM. Synthesis of 8-Oxa analogues of norcocaine endowed with interesting cocaine-like activity. Bioorganic & Medicinal Chemistry Letters. 9: 1831-6. PMID 10406650 DOI: 10.1016/S0960-894X(99)00273-5 |
0.477 |
|
| 1999 |
Simoni D, Roberti M, Rondanin R, Kozikowski AP. Enantioselective deprotonation of the 8-oxabicyclo[3.2.1]octan-3-one: Synthesis of 8-oxa-norcocaines and 8-oxa-pseudonorcocaines Tetrahedron Letters. 40: 4425-4428. DOI: 10.1016/S0040-4039(99)00763-7 |
0.488 |
|
| 1998 |
Garuti L, Roberti M, Rossi T, Castelli M, Malagoli M. Synthesis and antiproliferative activity of 3-substituted 1H-indole [3,2-d]-l,2,3-triazin-4 (3H)-ones European Journal of Medicinal Chemistry. 33: 43-46. DOI: 10.1016/S0223-5234(99)80074-9 |
0.372 |
|
| 1996 |
Kozikowski AP, Simoni D, Manfredini S, Roberti M, Stoelwinder J. Synthesis of the 6- and 7-hydroxylated cocaines and pseudococaines Tetrahedron Letters. 37: 5333-5336. DOI: 10.1016/0040-4039(96)01123-9 |
0.465 |
|
| 1995 |
Garuti L, Roberti M, Rossi M, Giovanninetti G. Some new 3-methoxy-5-methyl-1,4-substituted pyrazoles Farmaco. 50: 815-818. PMID 8593179 |
0.309 |
|
| 1993 |
Pellicciari R, Natalini B, Costantino G, Garzon A, Luneia R, Mahmoud MR, Marinozzi M, Roberti M, Rosato GC, Shiba SA. Heterocyclic modulators of the NMDA receptor. Farmaco (Societã Chimica Italiana : 1989). 48: 151-7. PMID 8494596 |
0.405 |
|
| 1992 |
Kozikowski AP, Roberti M, Xiang L, Bergmann JS, Callahan PM, Cunningham KA, Johnson KM. Structure-activity relationship studies of cocaine: replacement of the C-2 ester group by vinyl argues against H-bonding and provides an esterase-resistant, high-affinity cocaine analogue. Journal of Medicinal Chemistry. 35: 4764-6. PMID 1469704 DOI: 10.1021/Jm00103A015 |
0.395 |
|
| 1992 |
Baraldi PG, Budriesi R, Cacciari B, Chiarini A, Garuti L, Giovanninetti G, Leoni A, Roberti M. Synthesis and Calcium Antagonist Activity of Dialkyl 1,4-Dihydro-2,6-dimethyl-4-(nitrogenous heteroaryl)-3,5-pyridine Dicarboxylates Collection of Czechoslovak Chemical Communications. 57: 169-178. DOI: 10.1135/Cccc19920169 |
0.356 |
|
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