Year |
Citation |
Score |
2020 |
Szlavik Z, Csekei M, Paczal A, Szabo ZB, Sipos S, Radics G, Proszenyak A, Balint B, Murray J, Davidson J, Chen I, Dokurno P, Surgenor AE, Daniels ZM, Hubbard RE, et al. Discovery of S64315, a Potent and Selective Mcl-1 Inhibitor. Journal of Medicinal Chemistry. PMID 33146521 DOI: 10.1021/acs.jmedchem.0c01234 |
0.368 |
|
2019 |
Szlávik Z, Ondi L, Csékei M, Paczal A, Szabó ZB, Radics G, Murray J, Davidson J, Chen I, Davis B, Hubbard RE, Pedder C, Dokurno P, Surgenor A, Smith J, et al. Structure-Guided Discovery of a Selective Mcl-1 Inhibitor with Cellular Activity. Journal of Medicinal Chemistry. PMID 31339316 DOI: 10.1021/Acs.Jmedchem.9B00134 |
0.394 |
|
2019 |
Maragno AL, Mistry P, Kotschy A, Szlavik Z, Murray J, Davidson J, Toumelin-Braizat GL, Chanrion M, Bruno A, Claperon A, Maacke H, Morris E, Wang Y, Derreal A, Csekei M, et al. Abstract 4482: S64315 (MIK665) is a potent and selective Mcl1 inhibitor with strong antitumor activity across a diverse range of hematologic tumor models Cancer Research. 79: 4482-4482. DOI: 10.1158/1538-7445.Am2019-4482 |
0.393 |
|
2018 |
Casara P, Davidson J, Claperon A, Le Toumelin-Braizat G, Vogler M, Bruno A, Chanrion M, Lysiak-Auvity G, Le Diguarher T, Starck JB, Chen I, Whitehead N, Graham C, Matassova N, Dokurno P, et al. S55746 is a novel orally active BCL-2 selective and potent inhibitor that impairs hematological tumor growth. Oncotarget. 9: 20075-20088. PMID 29732004 DOI: 10.18632/oncotarget.24744 |
0.391 |
|
2018 |
Casara P, Davidson J, Claperon A, Toumelin-Braizat GL, Vogler M, Bruno A, Chanrion M, Lysiak-Auvity G, Diguarher TL, Starck J-, Chen I, Whitehead N, Graham C, Matassova N, Dokurno P, et al. S55746 is a novel orally active BCL-2 selective and potent inhibitor that impairs hematological tumor growth. Oncotarget. 9: 20075-20088. DOI: 10.2210/Pdb6Gl8/Pdb |
0.397 |
|
2016 |
Kotschy A, Szlavik Z, Murray J, Davidson J, Maragno AL, Le Toumelin-Braizat G, Chanrion M, Kelly GL, Gong JN, Moujalled DM, Bruno A, Csekei M, Paczal A, Szabo ZB, Sipos S, et al. The MCL1 inhibitor S63845 is tolerable and effective in diverse cancer models. Nature. PMID 27760111 DOI: 10.1038/Nature19830 |
0.377 |
|
2012 |
Geneste O, Murray J, Diguarher TL, Starck J, Casara P, Nanteuil GD, Davidson J, Nunns C, Graham C, Matassova N, Chen I, Whitehead N, Dokurno P, Bruno A, Pierré A, et al. Abstract 2782: Bcl-2 selective antagonists show antitumor activity without dose limiting platelet toxicity Cancer Research. 72: 2782-2782. DOI: 10.1158/1538-7445.Am2012-2782 |
0.4 |
|
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